Entity Details

Primary name GLP1R_HUMAN
Entity type UniProt
Source Source Link

Details

AccessionP43220
EntryNameGLP1R_HUMAN
FullNameGlucagon-like peptide 1 receptor
TaxID9606
Evidenceevidence at protein level
Length463
SequenceStatuscomplete
DateCreated1995-11-01
DateModified2021-06-02

Ontological Relatives

GenesGLP1R

GO terms

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GOName
GO:0002862 negative regulation of inflammatory response to antigenic stimulus
GO:0004888 transmembrane signaling receptor activity
GO:0004967 glucagon receptor activity
GO:0005886 plasma membrane
GO:0005887 integral component of plasma membrane
GO:0007166 cell surface receptor signaling pathway
GO:0007186 G protein-coupled receptor signaling pathway
GO:0007188 adenylate cyclase-modulating G protein-coupled receptor signaling pathway
GO:0007189 adenylate cyclase-activating G protein-coupled receptor signaling pathway
GO:0007190 activation of adenylate cyclase activity
GO:0007204 positive regulation of cytosolic calcium ion concentration
GO:0008528 G protein-coupled peptide receptor activity
GO:0016021 integral component of membrane
GO:0017046 peptide hormone binding
GO:0019933 cAMP-mediated signaling
GO:0044508 glucagon-like peptide 1 receptor activity
GO:0045777 positive regulation of blood pressure
GO:0050796 regulation of insulin secretion

Subcellular Location

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Subcellular Location
Cell membrane

Domains

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DomainNameCategoryType
IPR000832 GPCR, family 2, secretin-likeFamilyFamily
IPR001879 GPCR, family 2, extracellular hormone receptor domainDomainDomain
IPR003290 GPCR, family 2, glucagon-like peptide-1/glucagon receptorFamilyFamily
IPR003292 GPCR, family 2, glucagon-like peptide-1 receptorFamilyFamily
IPR017981 GPCR, family 2-likeDomainDomain
IPR017983 GPCR, family 2, secretin-like, conserved siteSiteConserved site
IPR036445 GPCR family 2, extracellular hormone receptor domain superfamilyFamilyHomologous superfamily

Diseases

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Drugs

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DrugNameSourceType
DB00040 GlucagonDrugbankbiotech
DB01276 ExenatideDrugbankbiotech
DB06655 LiraglutideDrugbankbiotech
DB09043 AlbiglutideDrugbankbiotech
DB09045 DulaglutideDrugbankbiotech
DB09265 LixisenatideDrugbanksmall molecule
DB13928 SemaglutideDrugbanksmall molecule

Interactions

124 interactions

InteractorPartnerSourcesPublicationsLink
GLP1R_HUMANKR107_HUMANBioGRID, IntAct25416956 details
GLP1R_HUMANKR108_HUMANBioGRID, IntAct25416956 details
GLP1R_HUMANNT2NA_HUMANBioGRID, IntAct25416956 32296183 details
GLP1R_HUMANKR109_HUMANBioGRID, IntAct25416956 details
GLP1R_HUMANNT2NC_HUMANBioGRID, IntAct25416956 32296183 details
GLP1R_HUMANKRA59_HUMANBioGRID, IntAct32296183 details
GLP1R_HUMANCRTP1_HUMANBioGRID, IntAct32296183 details
GLP1R_HUMANKRA11_HUMANBioGRID, IntAct32296183 details
GLP1R_HUMANKR171_HUMANBioGRID, IntAct32296183 details
GLP1R_HUMANGLUC_HUMANBioGRID, HPRD11116211 18248821 details
GLP1R_HUMANACSF3_HUMANBioGRID23864651 details
GLP1R_HUMANAP2M1_HUMANBioGRID23864651 details
GLP1R_HUMANAPH1A_HUMANBioGRID23864651 details
GLP1R_HUMANAPLP1_HUMANBioGRID23864651 details
GLP1R_HUMANARFRP_HUMANBioGRID23864651 details
GLP1R_HUMANAT131_HUMANBioGRID23864651 details
GLP1R_HUMANVATO_HUMANBioGRID23864651 details
GLP1R_HUMANRTRAF_HUMANBioGRID23864651 details
GLP1R_HUMANCR032_HUMANBioGRID23864651 details
GLP1R_HUMANCYTM1_HUMANBioGRID23864651 details
GLP1R_HUMANCAND2_HUMANBioGRID23864651 details
GLP1R_HUMANCD81_HUMANBioGRID23864651 28597972 details
GLP1R_HUMANCEND_HUMANBioGRID23864651 details
GLP1R_HUMANCFAI_HUMANBioGRID23864651 details
GLP1R_HUMANELOV1_HUMANBioGRID23864651 details
GLP1R_HUMANERP29_HUMANBioGRID23864651 details
GLP1R_HUMANFDFT_HUMANBioGRID23864651 details
GLP1R_HUMANGABR2_HUMANBioGRID23864651 details
GLP1R_HUMANGPR37_HUMANBioGRID23864651 details
GLP1R_HUMANHEPS_HUMANBioGRID23864651 details
GLP1R_HUMANIFM3_HUMANBioGRID23864651 26272612 details
GLP1R_HUMANMFSD5_HUMANBioGRID23864651 details
GLP1R_HUMANRM22_HUMANBioGRID23864651 details
GLP1R_HUMANMYL6_HUMANBioGRID23864651 details
GLP1R_HUMANNEUG_HUMANBioGRID23864651 details
GLP1R_HUMANNUCKS_HUMANBioGRID23864651 details
GLP1R_HUMANPAQR6_HUMANBioGRID23864651 details
GLP1R_HUMANP4HTM_HUMANBioGRID23864651 details
GLP1R_HUMANPIGG_HUMANBioGRID23864651 details
GLP1R_HUMANS15A4_HUMANBioGRID23864651 28597972 details
GLP1R_HUMANCOPT2_HUMANBioGRID23864651 details
GLP1R_HUMANSTMN1_HUMANBioGRID23864651 details
GLP1R_HUMANSTMN3_HUMANBioGRID23864651 details
GLP1R_HUMANSTML2_HUMANBioGRID23864651 details
GLP1R_HUMANSVOP_HUMANBioGRID23864651 details
GLP1R_HUMANSNG3_HUMANBioGRID23864651 details
GLP1R_HUMANTM147_HUMANBioGRID23864651 details
GLP1R_HUMANTSN13_HUMANBioGRID23864651 details
GLP1R_HUMANKR103_HUMANBioGRID25416956 details
GLP1R_HUMANBI1_HUMANBioGRID26272612 details
GLP1R_HUMANCLIP4_HUMANBioGRID26272612 details
GLP1R_HUMANCEL3B_HUMANBioGRID26272612 details
GLP1R_HUMANCLD7_HUMANBioGRID26272612 details
GLP1R_HUMANCC167_HUMANBioGRID26272612 details
GLP1R_HUMANCOL_HUMANBioGRID26272612 details
GLP1R_HUMANDAD1_HUMANBioGRID26272612 details
GLP1R_HUMANGNAS3_HUMANBioGRID26272612 details
GLP1R_HUMANGNAS2_HUMANBioGRID26272612 details
GLP1R_HUMANALEX_HUMANBioGRID26272612 details
GLP1R_HUMANGNAS1_HUMANBioGRID26272612 details
GLP1R_HUMANSG2A1_HUMANBioGRID26272612 details
GLP1R_HUMANMTCH2_HUMANBioGRID26272612 details
GLP1R_HUMANGP2_HUMANBioGRID26272612 details
GLP1R_HUMANAMD_HUMANBioGRID26272612 details
GLP1R_HUMANGP108_HUMANBioGRID26272612 details
GLP1R_HUMANRTN4_HUMANBioGRID26272612 details
GLP1R_HUMANSC11C_HUMANBioGRID26272612 details
GLP1R_HUMANSNG4_HUMANBioGRID26272612 details
GLP1R_HUMANT4S4_HUMANBioGRID26272612 details
GLP1R_HUMANTMCO3_HUMANBioGRID26272612 details
GLP1R_HUMANTRY2_HUMANBioGRID26272612 details
GLP1R_HUMANCD003_HUMANBioGRID26272612 details
GLP1R_HUMANAIG1_HUMANBioGRID26272612 details
GLP1R_HUMANOST4_HUMANBioGRID26272612 details
GLP1R_HUMANEMP2_HUMANBioGRID26272612 details
GLP1R_HUMANNU4LM_HUMANBioGRID26272612 details
GLP1R_HUMANCNIH4_HUMANBioGRID26272612 details
GLP1R_HUMANRENR_HUMANBioGRID26272612 details
GLP1R_HUMANRTN3_HUMANBioGRID26272612 details
GLP1R_HUMANSELK_HUMANBioGRID26272612 details
GLP1R_HUMANTOM6_HUMANBioGRID26272612 details
GLP1R_HUMANSYS1_HUMANBioGRID28597972 details
GLP1R_HUMANIEX1_HUMANBioGRID28597972 details
GLP1R_HUMANSPTSA_HUMANBioGRID28597972 details
GLP1R_HUMANSPYA_HUMANBioGRID28597972 details
GLP1R_HUMANSAA1_HUMANBioGRID28597972 details
GLP1R_HUMANT176B_HUMANBioGRID28597972 details
GLP1R_HUMANUD19_HUMANBioGRID28597972 details
GLP1R_HUMANA1AT_HUMANBioGRID28597972 details
GLP1R_HUMANFRIL_HUMANBioGRID28597972 details
GLP1R_HUMANLAP4A_HUMANBioGRID28597972 details
GLP1R_HUMANEMC7_HUMANBioGRID28597972 details
GLP1R_HUMANZNF99_HUMANBioGRID28597972 details
GLP1R_HUMANEBP_HUMANBioGRID28597972 details
GLP1R_HUMANATP6_HUMANBioGRID28597972 details
GLP1R_HUMANAT5G3_HUMANBioGRID28597972 details
GLP1R_HUMANCD63_HUMANBioGRID28597972 details
GLP1R_HUMANSERP1_HUMANBioGRID28597972 details
GLP1R_HUMANVAPB_HUMANBioGRID28597972 details
GLP1R_HUMANPSMD8_HUMANBioGRID28597972 details
GLP1R_HUMANASGR2_HUMANBioGRID28597972 details
GLP1R_HUMANCOMT_HUMANBioGRID28597972 details
GLP1R_HUMANDHRS7_HUMANBioGRID28597972 details
GLP1R_HUMANRNF5_HUMANBioGRID28597972 details
GLP1R_HUMANFGL1_HUMANBioGRID28597972 details
GLP1R_HUMANCXB1_HUMANBioGRID28597972 details
GLP1R_HUMANG6PT1_HUMANBioGRID28597972 details
GLP1R_HUMANHEPC_HUMANBioGRID28597972 details
GLP1R_HUMANKHK_HUMANBioGRID28597972 details
GLP1R_HUMANOCAD2_HUMANBioGRID28597972 details
GLP1R_HUMANPPIB_HUMANBioGRID28597972 details
GLP1R_HUMANLFG1_HUMANBioGRID28597972 details
GLP1R_HUMANPOMT2_HUMANBioGRID28597972 details
GLP1R_HUMANRAB5B_HUMANBioGRID25044020 details
GLP1R_HUMANRAB5C_HUMANBioGRID25044020 details
GLP1R_HUMANPGRC1_HUMANBioGRID25044020 details
GLP1R_HUMANCAV1_HUMANBioGRID25044020 details
GLP1R_HUMANKRA13_HUMANBioGRID32296183 details
GLP1R_HUMANCALM2_HUMANHPRD, MINT15670850 details
GLP1R_HUMANARRB1_HUMANDIP18445652 details
GLP1R_HUMANSUMO1_HUMANBioGRID22234371 details
GLP1R_HUMANCALM1_HUMANHPRD15670850 details
GLP1R_HUMANCALM3_HUMANHPRD15670850 details
GLP1R_HUMANGASP1_HUMANHPRD15452121 details