Entity Details

Primary name ACM3_HUMAN
Entity type UniProt
Source Source Link

Details

AccessionP20309
EntryNameACM3_HUMAN
FullNameMuscarinic acetylcholine receptor M3
TaxID9606
Evidenceevidence at protein level
Length590
SequenceStatuscomplete
DateCreated1991-02-01
DateModified2021-06-02

Ontological Relatives

GenesCHRM3

GO terms

Show/Hide Table
GOName
GO:0003056 regulation of vascular associated smooth muscle contraction
GO:0004435 phosphatidylinositol phospholipase C activity
GO:0004993 G protein-coupled serotonin receptor activity
GO:0005789 endoplasmic reticulum membrane
GO:0005886 plasma membrane
GO:0005887 integral component of plasma membrane
GO:0006464 cellular protein modification process
GO:0007165 signal transduction
GO:0007186 G protein-coupled receptor signaling pathway
GO:0007187 G protein-coupled receptor signaling pathway, coupled to cyclic nucleotide second messenger
GO:0007197 adenylate cyclase-inhibiting G protein-coupled acetylcholine receptor signaling pathway
GO:0007213 G protein-coupled acetylcholine receptor signaling pathway
GO:0007268 chemical synaptic transmission
GO:0007399 nervous system development
GO:0009925 basal plasma membrane
GO:0016323 basolateral plasma membrane
GO:0016907 G protein-coupled acetylcholine receptor activity
GO:0019722 calcium-mediated signaling
GO:0030425 dendrite
GO:0030594 neurotransmitter receptor activity
GO:0032412 regulation of ion transmembrane transporter activity
GO:0038023 signaling receptor activity
GO:0042166 acetylcholine binding
GO:0045202 synapse
GO:0045211 postsynaptic membrane
GO:0045987 positive regulation of smooth muscle contraction
GO:0046541 saliva secretion
GO:0095500 acetylcholine receptor signaling pathway

Subcellular Location

Show/Hide Table
Subcellular Location
Basolateral cell membrane
Cell junction
Cell membrane
Endoplasmic reticulum membrane

Domains

Show/Hide Table
DomainNameCategoryType
IPR000276 G protein-coupled receptor, rhodopsin-likeFamilyFamily
IPR000995 Muscarinic acetylcholine receptor familyFamilyFamily
IPR001183 Muscarinic acetylcholine receptor M3FamilyFamily
IPR017452 GPCR, rhodopsin-like, 7TMDomainDomain

Diseases

Show/Hide Table

Drugs

Show/Hide Table
DrugNameSourceType
DB00185 CevimelineDrugbanksmall molecule
DB00193 TramadolDrugbanksmall molecule
DB00202 SuccinylcholineDrugbanksmall molecule
DB00209 TrospiumDrugbanksmall molecule
DB00246 ZiprasidoneDrugbanksmall molecule
DB00280 DisopyramideDrugbanksmall molecule
DB00321 AmitriptylineDrugbanksmall molecule
DB00332 IpratropiumDrugbanksmall molecule
DB00334 OlanzapineDrugbanksmall molecule
DB00340 MetixeneDrugbanksmall molecule
DB00342 TerfenadineDrugbanksmall molecule
DB00363 ClozapineDrugbanksmall molecule
DB00366 DoxylamineDrugbanksmall molecule
DB00376 TrihexyphenidylDrugbanksmall molecule
DB00383 OxyphencyclimineDrugbanksmall molecule
DB00387 ProcyclidineDrugbanksmall molecule
DB00408 LoxapineDrugbanksmall molecule
DB00411 CarbamoylcholineDrugbanksmall molecule
DB00424 HyoscyamineDrugbanksmall molecule
DB00434 CyproheptadineDrugbanksmall molecule
DB00454 MeperidineDrugbanksmall molecule
DB00458 ImipramineDrugbanksmall molecule
DB00462 Methscopolamine bromideDrugbanksmall molecule
DB00477 ChlorpromazineDrugbanksmall molecule
DB00496 DarifenacinDrugbanksmall molecule
DB00502 HaloperidolDrugbanksmall molecule
DB00505 TridihexethylDrugbanksmall molecule
DB00517 Anisotropine methylbromideDrugbanksmall molecule
DB00540 NortriptylineDrugbanksmall molecule
DB00543 AmoxapineDrugbanksmall molecule
DB00568 CinnarizineDrugbanksmall molecule
DB00572 AtropineDrugbanksmall molecule
DB00599 ThiopentalDrugbanksmall molecule
DB00622 NicardipineDrugbanksmall molecule
DB00715 ParoxetineDrugbanksmall molecule
DB00725 Homatropine methylbromideDrugbanksmall molecule
DB00726 TrimipramineDrugbanksmall molecule
DB00747 ScopolamineDrugbanksmall molecule
DB00767 BenzquinamideDrugbanksmall molecule
DB00777 PropiomazineDrugbanksmall molecule
DB00809 TropicamideDrugbanksmall molecule
DB00835 BrompheniramineDrugbanksmall molecule
DB00934 MaprotilineDrugbanksmall molecule
DB00940 MethanthelineDrugbanksmall molecule
DB00986 GlycopyrroniumDrugbanksmall molecule
DB01019 BethanecholDrugbanksmall molecule
DB01036 TolterodineDrugbanksmall molecule
DB01062 OxybutyninDrugbanksmall molecule
DB01069 PromethazineDrugbanksmall molecule
DB01085 PilocarpineDrugbanksmall molecule
DB01142 DoxepinDrugbanksmall molecule
DB01151 DesipramineDrugbanksmall molecule
DB01221 KetamineDrugbanksmall molecule
DB01224 QuetiapineDrugbanksmall molecule
DB01226 MivacuriumDrugbanksmall molecule
DB01231 DiphenidolDrugbanksmall molecule
DB01238 AripiprazoleDrugbanksmall molecule
DB01239 ChlorprothixeneDrugbanksmall molecule
DB01337 PancuroniumDrugbanksmall molecule
DB01338 PipecuroniumDrugbanksmall molecule
DB01403 MethotrimeprazineDrugbanksmall molecule
DB01409 TiotropiumDrugbanksmall molecule
DB01591 SolifenacinDrugbanksmall molecule
DB01625 IsopropamideDrugbanksmall molecule
DB03128 AcetylcholineDrugbanksmall molecule
DB04365 ArecolineDrugbanksmall molecule
DB04843 MepenzolateDrugbanksmall molecule
DB05752 ALKS 27Drugbanksmall molecule
DB06153 PizotifenDrugbanksmall molecule
DB06702 FesoterodineDrugbanksmall molecule
DB06709 MethacholineDrugbanksmall molecule
DB06787 HexocycliumDrugbanksmall molecule
DB08897 AclidiniumDrugbanksmall molecule
DB09076 UmeclidiniumDrugbanksmall molecule
DB09089 TrimebutineDrugbanksmall molecule
DB09167 DosulepinDrugbanksmall molecule
DB09194 EtoperidoneDrugbanksmall molecule
DB09262 ImidafenacinDrugbanksmall molecule
DB09300 ButylscopolamineDrugbanksmall molecule
DB11181 HomatropineDrugbanksmall molecule
DB11235 ThonzylamineDrugbanksmall molecule
DB11855 RevefenacinDrugbanksmall molecule
DB12278 PropiverineDrugbanksmall molecule
DB13581 RociverineDrugbanksmall molecule
DB13720 DiphemanilDrugbanksmall molecule
DB14185 Aripiprazole lauroxilDrugbanksmall molecule

Interactions

35 interactions

InteractorPartnerSourcesPublicationsLink
ACM3_HUMANBASI_HUMANBioGRID, MINT28298427 details
ACM3_HUMANCD2B2_HUMANBioGRID, MINT28298427 details
ACM3_HUMANRCAF1_HUMANBioGRID, MINT28298427 details
ACM3_HUMANCOMD7_HUMANBioGRID, MINT28298427 details
ACM3_HUMANGNAS2_HUMANBioGRID, MINT28298427 details
ACM3_HUMANJKIP1_HUMANBioGRID, MINT28298427 details
ACM3_HUMANMAGD2_HUMANBioGRID, MINT28298427 details
ACM3_HUMANP121C_HUMANMINT28298427 details
ACM3_HUMANSEPT3_HUMANBioGRID, MINT28298427 details
ACM3_HUMANCC184_HUMANBioGRID, MINT28298427 details
ACM3_HUMANSGSM3_HUMANBioGRID, MINT28298427 details
ACM3_HUMANTAP1_HUMANBioGRID, MINT28298427 details
ACM3_HUMANTPM3_HUMANBioGRID, MINT28298427 details
ACM3_HUMANYIPF3_HUMANBioGRID, MINT28298427 details
ACM3_HUMANACM5_HUMANIntAct20398705 details
ACM3_HUMANACM3_HUMANIntAct20398705 details
ACM3_HUMANARF1_HUMANBioGRID, HPRD12799371 details
ACM3_HUMANARF6_HUMANBioGRID, HPRD12799371 details
ACM3_HUMANKC1A_HUMANBioGRID, HPRD10777483 details
ACM3_HUMANSET_HUMANBioGRID17065150 details
ACM3_HUMANRGS7_HUMANBioGRID19182865 details
ACM3_HUMANCALM1_HUMANBioGRID28298427 details
ACM3_HUMANCALM2_HUMANBioGRID28298427 details
ACM3_HUMANCALM3_HUMANBioGRID28298427 details
ACM3_HUMANGNAS3_HUMANBioGRID28298427 details
ACM3_HUMANALEX_HUMANBioGRID28298427 details
ACM3_HUMANGNAS1_HUMANBioGRID28298427 details
ACM3_HUMANNEB2_HUMANHPRD, MINT17464283 details
ACM3_HUMANNALCN_HUMANMINT19575010 details
ACM3_HUMANMDM2_HUMANIntAct20195357 details
ACM3_HUMANRGS4_HUMANDIP20385802 details
ACM3_HUMANGRAB_HUMANHPRD11665980 details
ACM3_HUMANGRK6_HUMANHPRD11856737 details
ACM3_HUMANGNAQ_HUMANHPRD7629074 details
ACM3_HUMANGASP1_HUMANHPRD15452121 details