Entity Details

Primary name GABR1_HUMAN
Entity type UniProt
Source Source Link

Details

AccessionQ9UBS5
EntryNameGABR1_HUMAN
FullNameGamma-aminobutyric acid type B receptor subunit 1
TaxID9606
Evidenceevidence at protein level
Length961
SequenceStatuscomplete
DateCreated2001-01-11
DateModified2021-06-02

Ontological Relatives

GenesGABBR1

GO terms

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GOName
GO:0004888 transmembrane signaling receptor activity
GO:0004965 G protein-coupled GABA receptor activity
GO:0005576 extracellular region
GO:0005737 cytoplasm
GO:0005886 plasma membrane
GO:0005887 integral component of plasma membrane
GO:0007186 G protein-coupled receptor signaling pathway
GO:0007193 adenylate cyclase-inhibiting G protein-coupled receptor signaling pathway
GO:0007214 gamma-aminobutyric acid signaling pathway
GO:0030425 dendrite
GO:0038039 G protein-coupled receptor heterodimeric complex
GO:0042734 presynaptic membrane
GO:0045211 postsynaptic membrane
GO:0098685 Schaffer collateral - CA1 synapse
GO:0098982 GABA-ergic synapse
GO:0099579 G protein-coupled neurotransmitter receptor activity involved in regulation of postsynaptic membrane potential
GO:0150099 neuron-glial cell signaling
GO:1901381 positive regulation of potassium ion transmembrane transport

Subcellular Location

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Subcellular Location
Cell junction
Cell membrane
Cell projection
Secreted

Domains

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DomainNameCategoryType
IPR000436 Sushi/SCR/CCP domainDomainDomain
IPR001828 Receptor, ligand binding regionDomainDomain
IPR002455 GPCR family 3, GABA-B receptorFamilyFamily
IPR002456 GPCR family 3, gamma-aminobutyric acid receptor, type B1FamilyFamily
IPR017978 GPCR family 3, C-terminalDomainDomain
IPR028082 Periplasmic binding protein-like IFamilyHomologous superfamily
IPR035976 Sushi/SCR/CCP superfamilyFamilyHomologous superfamily

Diseases

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Drugs

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DrugNameSourceType
DB00181 BaclofenDrugbanksmall molecule
DB00837 ProgabideDrugbanksmall molecule
DB01956 TaurineDrugbanksmall molecule
DB02530 gamma-Aminobutyric acidDrugbanksmall molecule
DB05010 SGS-742Drugbanksmall molecule
DB06354 TezampanelDrugbanksmall molecule
DB08891 ArbaclofenDrugbanksmall molecule
DB08892 Arbaclofen PlacarbilDrugbanksmall molecule

Interactions

31 interactions

InteractorPartnerSourcesPublicationsLink
GABR1_HUMANCHFR_HUMANHPRD, IntAct16169070 details
GABR1_HUMANNSF_HUMANHPRD, MINT16724110 details
GABR1_HUMANGABR2_HUMANBioGRID, DIP, HPRD, IntAct, MINT10075644 16724110 24305054 24658140 26817839 30971491 32555460 32580208 32581365 9872316 details
GABR1_HUMANABL1_HUMANIntAct17474147 details
GABR1_HUMANCRK_HUMANIntAct17474147 details
GABR1_HUMANFYN_HUMANIntAct17474147 details
GABR1_HUMANGRB2_HUMANIntAct17474147 details
GABR1_HUMANNCK1_HUMANIntAct17474147 details
GABR1_HUMANP85A_HUMANIntAct17474147 details
GABR1_HUMANMAX_HUMANBioGRID, IntAct20195357 details
GABR1_HUMANGPR37_HUMANBioGRID, MINT28298427 details
GABR1_HUMANBKRB1_HUMANBioGRID, MINT28298427 details
GABR1_HUMANCCR8_HUMANBioGRID, MINT28298427 details
GABR1_HUMANDRD2_HUMANBioGRID, MINT28298427 details
GABR1_HUMANSMO_HUMANBioGRID, MINT28298427 details
GABR1_HUMANGABR1_HUMANDIP32580208 details
GABR1_HUMANJKIP1_HUMANBioGRID, HPRD14718537 details
GABR1_HUMANATF5_HUMANBioGRID, HPRD11087824 details
GABR1_HUMANATF4_HUMANBioGRID11087824 details
GABR1_HUMANGNAO_HUMANBioGRID17185339 details
GABR1_HUMANKCNJ6_HUMANBioGRID17185339 details
GABR1_HUMANRGS4_HUMANBioGRID17185339 details
GABR1_HUMANCPEB2_HUMANBioGRID22157746 details
GABR1_HUMAN1433Z_HUMANHPRD11178869 details
GABR1_HUMANUBP14_HUMANBioGRID26817839 details
GABR1_HUMANDDIT3_HUMANBioGRID16081421 details
GABR1_HUMANKCD16_HUMANBioGRID30971491 details
GABR1_HUMANKCNJ3_HUMANBioGRID16809021 details
GABR1_HUMANGBB1_HUMANBioGRID16809021 details
GABR1_HUMANGBG2_HUMANBioGRID16809021 details
GABR1_HUMANCASR_HUMANBioGRID17591780 details