Entity Details

Primary name GRIA1_HUMAN
Entity type UniProt
Source Source Link

Details

AccessionP42261
EntryNameGRIA1_HUMAN
FullNameGlutamate receptor 1
TaxID9606
Evidenceevidence at protein level
Length906
SequenceStatuscomplete
DateCreated1995-11-01
DateModified2021-06-02

Ontological Relatives

GenesGRIA1

GO terms

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GOName
GO:0001540 amyloid-beta binding
GO:0004971 AMPA glutamate receptor activity
GO:0005789 endoplasmic reticulum membrane
GO:0005886 plasma membrane
GO:0006888 endoplasmic reticulum to Golgi vesicle-mediated transport
GO:0007165 signal transduction
GO:0007268 chemical synaptic transmission
GO:0007616 long-term memory
GO:0008066 glutamate receptor activity
GO:0009986 cell surface
GO:0012507 ER to Golgi transport vesicle membrane
GO:0014069 postsynaptic density
GO:0015276 ligand-gated ion channel activity
GO:0030165 PDZ domain binding
GO:0030425 dendrite
GO:0030666 endocytic vesicle membrane
GO:0030672 synaptic vesicle membrane
GO:0031623 receptor internalization
GO:0031901 early endosome membrane
GO:0032281 AMPA glutamate receptor complex
GO:0032591 dendritic spine membrane
GO:0033116 endoplasmic reticulum-Golgi intermediate compartment membrane
GO:0038023 signaling receptor activity
GO:0043025 neuronal cell body
GO:0043197 dendritic spine
GO:0044308 axonal spine
GO:0044309 neuron spine
GO:0048208 COPII vesicle coating
GO:0055037 recycling endosome
GO:0055038 recycling endosome membrane
GO:0060076 excitatory synapse
GO:0060292 long-term synaptic depression
GO:0071242 cellular response to ammonium ion
GO:0097060 synaptic membrane
GO:0098978 glutamatergic synapse
GO:0099061 integral component of postsynaptic density membrane
GO:0099544 perisynaptic space
GO:0099583 neurotransmitter receptor activity involved in regulation of postsynaptic cytosolic calcium ion concentration
GO:1904315 transmitter-gated ion channel activity involved in regulation of postsynaptic membrane potential
GO:2000310 regulation of NMDA receptor activity

Subcellular Location

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Subcellular Location
Cell junction
Cell membrane
Cell projection
Early endosome membrane
Endoplasmic reticulum membrane
Recycling endosome membrane

Domains

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DomainNameCategoryType
IPR001320 Ionotropic glutamate receptorDomainDomain
IPR001508 Ionotropic glutamate receptor, metazoaFamilyFamily
IPR001828 Receptor, ligand binding regionDomainDomain
IPR019594 Ionotropic glutamate receptor, L-glutamate and glycine-binding domainDomainDomain
IPR028082 Periplasmic binding protein-like IFamilyHomologous superfamily

Diseases

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Drugs

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DrugNameSourceType
DB00142 Glutamic acidDrugbanksmall molecule
DB00237 ButabarbitalDrugbanksmall molecule
DB00555 LamotrigineDrugbanksmall molecule
DB00753 IsofluraneDrugbanksmall molecule
DB00898 EthanolDrugbanksmall molecule
DB01028 MethoxyfluraneDrugbanksmall molecule
DB01189 DesfluraneDrugbanksmall molecule
DB01236 SevofluraneDrugbanksmall molecule
DB04982 TalampanelDrugbanksmall molecule
DB05047 CX-717Drugbanksmall molecule
DB06247 CX516Drugbanksmall molecule
DB08883 PerampanelDrugbanksmall molecule
DB09289 TianeptineDrugbanksmall molecule
DB13146 Fluciclovine (18F)Drugbanksmall molecule

Interactions

40 interactions

InteractorPartnerSourcesPublicationsLink
GRIA1_HUMANKAPCA_HUMANHPRD, MINT8663994 details
GRIA1_HUMANPP1A_HUMANDIP20305656 details
GRIA1_HUMANASCL4_HUMANIntAct32814053 details
GRIA1_HUMANKLF15_HUMANIntAct32814053 details
GRIA1_HUMANRB11B_HUMANIntAct32814053 details
GRIA1_HUMANBECN1_HUMANIntAct32814053 details
GRIA1_HUMANZN232_HUMANIntAct32814053 details
GRIA1_HUMANE41L2_HUMANBioGRID, HPRD11050113 details
GRIA1_HUMANDLG1_HUMANBioGRID, HPRD11567040 12933808 23864692 9677374 details
GRIA1_HUMANPICK1_HUMANBioGRID, HPRD11891216 details
GRIA1_HUMANGRIP1_HUMANBioGRID11891216 details
GRIA1_HUMANSDCB1_HUMANBioGRID, HPRD11891216 details
GRIA1_HUMANE41L1_HUMANBioGRID, HPRD11050113 12574408 details
GRIA1_HUMANUBP46_HUMANBioGRID26077708 details
GRIA1_HUMANSQSTM_HUMANBioGRID, HPRD19004011 26187466 details
GRIA1_HUMANNED4L_HUMANBioGRID28212375 details
GRIA1_HUMANKCC2A_HUMANBioGRID24706758 details
GRIA1_HUMANKPCA_HUMANBioGRID, HPRD24706758 8663994 details
GRIA1_HUMANKS6B1_HUMANBioGRID24706758 details
GRIA1_HUMANCXCR2_HUMANBioGRID, HPRD, MINT12507773 12888558 18508130 details
GRIA1_HUMANGRID2_HUMANBioGRID, HPRD12573530 details
GRIA1_HUMANCCG2_HUMANBioGRID, HPRD11140673 details
GRIA1_HUMANGRIA2_HUMANBioGRID10358037 14602821 18311135 24706758 details
GRIA1_HUMANGRIK2_HUMANBioGRID, HPRD10358037 8288598 details
GRIA1_HUMANGRIA4_HUMANBioGRID, HPRD9466455 details
GRIA1_HUMANNEDD4_HUMANBioGRID21148011 21338354 details
GRIA1_HUMANANC2_HUMANBioGRID21186356 details
GRIA1_HUMANFZR1_HUMANBioGRID21186356 details
GRIA1_HUMANMYO5A_HUMANBioGRID18311135 details
GRIA1_HUMANRB11A_HUMANBioGRID18311135 details
GRIA1_HUMANHNRPQ_HUMANBioGRID20131911 details
GRIA1_HUMANGRIA3_HUMANBioGRID12700243 details
GRIA1_HUMANCASP8_HUMANHPRD11751897 details
GRIA1_HUMANCALX_HUMANHPRD10461883 details
GRIA1_HUMANBIP_HUMANHPRD10461883 details
GRIA1_HUMANGRIA1_HUMANHPRD11891216 details
GRIA1_HUMANGRAP1_HUMANHPRD10896157 details
GRIA1_HUMANHOME1_HUMANHPRD11418862 9069287 9808458 details
GRIA1_HUMANTRPC1_HUMANHPRD14614461 details
GRIA1_HUMANTANC1_HUMANHPRD15673434 details